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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T29174 | YIL781 hydrochloride | YIL 781,YIL-781,YIL781 HCl,YIL781 | |
YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM). | |||
T23543 | YIL 781 | GHSR | |
YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM). YIL 781 improves glucose homeostasis in vivo and in vitro by blocking ghrelin secretion... |